Li · Journal of controlled release : official journal of the Controlled Release Society 2025 · Preclinical laboratory and mechanistic study · n=?

Hyperbaric oxygen augments Doxil antitumor efficacy by reducing tumor-induced lactate.

Level 5 - mechanism / opinion, no new human data

Preclinical laboratory and mechanistic research with no human data

PubMed 40889529 · doi:10.1016/j.jconrel.2025.114181 · record verified 2026-08-26

What was done

Researchers investigated how tumor-elevated lactate affects the hepatic clearance of the nanomedicine Doxil and whether hyperbaric oxygen intervention could mitigate this clearance mechanism to improve antitumor efficacy. The study evaluated the impact of hyperbaric oxygen on tissue glycolysis, lactate levels, Kupffer cell M2 polarization, hepatic Doxil uptake, circulation time, and antitumor response.

What was found

The abstract reports no quantitative values or statistical metrics. Qualitatively, tumor-derived lactate was reported to accelerate Doxil clearance by driving M2 polarization in Kupffer cells. Hyperbaric oxygen countered this by suppressing glycolysis and reducing lactate levels in tumors and normal tissues, which diminished M2 Kupffer cell polarization, reduced hepatic Doxil uptake, prolonged blood circulation time, and enhanced antitumor efficacy.

Why it matters

This work identifies a metabolic mechanism whereby tumor-derived lactate accelerates nanomedicine clearance and highlights hyperbaric oxygen as a potential strategy to improve liposomal drug delivery.

Limits

The abstract provides no sample sizes, numerical data, effect sizes, or specific model details. Findings are derived from preclinical mechanistic research with no human clinical validation.